Profadol

Profadol (CI-572) is an opioid analgesic which was developed in the 1960s by Parke-Davis.[1] It acts as a mixed agonist-antagonist of the μ-opioid receptor. The analgetic potency is about the same as of pethidine (meperidine), the antagonistic effect is 1/50 of nalorphine.[2]

Not to be confused with propanol, propofol, or propranolol.
Profadol
Clinical data
ATC code
  • none
Legal status
Legal status
  • US: Analogue to a Schedule I/II drug (Analogue of Tapentadol, Schedule II)
Identifiers
CAS Number
PubChem CID
ChemSpider
UNII
ChEMBL
Chemical and physical data
FormulaC14H21NO
Molar mass219.32 g/mol g·mol−1

See also

References
  1. DE Patent 1303096
  2. Eberhard Schröder, Clemens Rufer, Ralph Schmiechen, Arzneimittelchemie I, Georg Thieme Verlag 1976 ISBN 3-13-520601-7
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