CUMYL-PINACA

CUMYL-PINACA
Legal status
Legal status	CA: Schedule II ; DE: NpSG (Industrial and scientific use only) ; UK: Under Psychoactive Substances Act ;
Identifiers
	IUPAC name 1-pentyl-N-(2-phenylpropan-2-yl)-1H-indazole-3-carboxamide;
CAS Number	1400742-15-5;
PubChem CID	86273676;
ChemSpider	48060412;
Chemical and physical data
Formula	C22H27N3O
Molar mass	349.5 g/mol g·mol−1
3D model (JSmol)	Interactive image;
	SMILES CCCCCN1N=C(C(=O)NC(C)(C)C2=CC=CC=C2)C2=CC=CC=C12;
	InChI InChI=1S/C22H27N3O/c1-4-5-11-16-25-19-15-10-9-14-18(19)20(24-25)21(26)23-22(2,3)17-12-7-6-8-13-17/h6-10,12-15H,4-5,11,16H2,1-3H3,(H,23,26); Key:LCBASRYREGWIJT-UHFFFAOYSA-N;

CUMYL-PINACA (also known as SGT-24) is an indazole-3-carboxamide based synthetic cannabinoid. CUMYL-PINACA acts as a potent agonist for the cannabinoid receptors, with approximately 3x selectivity for CB₁, having an EC₅₀ of 0.15nM for human CB₁ receptors and 0.41nM for human CB₂ receptors.[1]

Legal status

Sweden's public health agency suggested classifying CUMYL-PINACA as a hazardous substance, on November 10, 2014.[2]

References

Dobaja M, Grenc D, Kozelj G, Brvar M (March 2017). "Occupational transdermal poisoning with synthetic cannabinoid cumyl-PINACA". Clinical Toxicology. 55 (3): 193–195. doi:10.1080/15563650.2016.1278224. PMID 28084855.
"Cannabinoider föreslås bli klassade som hälsofarlig vara". Retrieved 11 July 2015.

This article is issued from Wikipedia. The text is licensed under Creative Commons - Attribution - Sharealike. Additional terms may apply for the media files.

[1] Dobaja M, Grenc D, Kozelj G, Brvar M (March 2017). "Occupational transdermal poisoning with synthetic cannabinoid cumyl-PINACA". Clinical Toxicology. 55 (3): 193–195. doi:10.1080/15563650.2016.1278224. PMID 28084855.

[2] "Cannabinoider föreslås bli klassade som hälsofarlig vara". Retrieved 11 July 2015.

CUMYL-PINACA

Legal status

See also

References