Olorinab

Olorinab (APD371) is a drug being developed by Arena Pharmaceuticals for the treatment of gastrointestinal pain associated with Crohn's disease and irritable bowel syndrome.[1] It acts as a potent and selective cannabinoid CB2 receptor agonist and is claimed to be orally active and peripherally selective.[2][3] Initial Phase IIa exploratory clinical trials have been successful,[4] with Phase IIb trials projected to start in 2019.[5]

Olorinab
Clinical data
Routes of
administration
Oral
Identifiers
CAS Number
PubChem CID
KEGG
Chemical and physical data
FormulaC18H24N5O3
Molar mass358.422 g·mol−1
3D model (JSmol)

See also

References

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