Apricoxib
Apricoxib is an experimental anticancer drug. It is a COX-2 inhibitor which is intended to improve standard therapy response in molecularly defined models of pancreatic cancer.[1] Development was abandoned in 2015 due to poor clinical trial results.[2]
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Formula | C19H20N2O3S |
Molar mass | 356.4387 g/mol g·mol−1 |
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See also
- Tilmacoxib
- cimicoxib
- NS-398
- Celecoxib
References
- Kirane, A. (2012). "Apricoxib, a Novel Inhibitor of COX-2, Markedly Improves Standard Therapy Response in Molecularly Defined Models of Pancreatic Cancer". Clinical Cancer Research. 18 (18): 5031–5042. doi:10.1158/1078-0432.CCR-12-0453. PMC 3777527. PMID 22829202.
- http://adisinsight.springer.com/drugs/800026002
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