Beta agonist

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β1 >> β2

β2 >> β1 (Beta-2 agonist)

Short-acting

  • Albuterol (ProAir HFA, Proventil, Ventolin HFA, ReliOn Ventolin HFA, Accuneb)
  • Terbutaline (Bricanyl)
  • Clenbuterol
  • Isoproterenol (β1 ≈ β2 )
  • Levosalbutamol, pirbuterol, procaterol, metaproterenol, fenoteol, bitolterol, ritodrine

Long-acting beta2 agonists

  • Clenbuterol
  • Salmeterol, formoterol (Symbicort), bambuterol, olodaterol, indacaterol (ultra-long-acting)

Nonselective Adrenergic Agonists

Authors

Claire