Bromazine
Bromazine (trade names Ambodryl[1], Ambrodil and others), also known as bromodiphenhydramine, is an antihistamine and anticholinergic.[2] It is a brominated form of diphenhydramine.
Not to be confused with Promazine.
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MedlinePlus | a682065 |
Routes of administration | Oral |
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Bioavailability | High |
Protein binding | 96% |
Metabolism | Mostly hepatic (CYP-mediated), also renal |
Elimination half-life | 1 to 4 hours |
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ECHA InfoCard | 100.003.854 |
Chemical and physical data | |
Formula | C17H20BrNO |
Molar mass | 334.251 g/mol g·mol−1 |
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References
- Baker, Charles E., Jr. (1974). Physicians' Desk Reference (28 ed.). Oradell, NJ 07649: Medical Economics Company. pp. 1076, 1081.
- MacLaren, W. R.; Bruff, W. C.; Eisenberg, B. C.; Weiner, H.; Martin, W. H. (1955). "A clinical comparison of carbinoxamine maleate, tripelennamine hydrochloride, and bromodiphenhydramine hydrochloride in treating allergic symptoms". Annals of Allergy. 13 (3): 307–312. PMID 14377226.
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See also: Receptor/signaling modulators • Monoamine metabolism modulators • Monoamine reuptake inhibitors |
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