Barbexaclone
Barbexaclone (Maliasin) is a salt compound of phenobarbital and levopropylhexedrine.[1] It was introduced in 1983. It has been reported to be as effective as phenobarbital but better tolerated; however, as of 2004, these "promising results"[2] had not yet been confirmed nor denied in controlled trials.
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| Phenobarbital | Barbiturate |
| Levopropylhexedrine | Stimulant (sympathomimetic) |
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| ECHA InfoCard | 100.022.278 |
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Potency
100 mg of barbexaclone is equivalent to 60 mg of phenobarbital.[1]
References
- Simon Shorvon; Emilio Perucca; Jerome Engel, Jr. (23 September 2015). The Treatment of Epilepsy. Wiley. pp. 1706–1707. ISBN 978-1-118-93699-3.
- Salles Barbosa, MF (September 1978). "[Barbexaclone in the treatment of cerebral dysrhythmia]". Arquivos de Neuro-Psiquiatria. 36 (3): 245–9. doi:10.1590/s0004-282x1978000300009. PMID 28716.
- Bibliography
- The Treatment of Epilepsy 2nd Ed by S. D. Shorvon (Editor), David R. Fish (Editor), Emilio Perucca (Editor), W. Edwin Dodson (Editor). Published by Blackwell 2004. p. 472. ISBN 0-632-06046-8
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See also: Receptor/signaling modulators • GABA receptor modulators • GABA metabolism/transport modulators | |
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